Aug 2026
Design, synthesis and dual anticancer and antibacterial evaluation of novel 1,3,4-oxadiazole-2-thiol derivatives targeting EGFR and DNA Gyrase B: integrated docking, DFT and ADMET studies.
1,3,4-oxadiazole-2-thiol derivatives are established as promising dual-action therapeutic scaffolds for anticancer and antibacterial activities through computational and experimental approaches.
Ila M. Ram, Jay B. Maheta, Darshna K. Lakhnotra et al.
· Future Medicinal Chemistry · 0 citations