Review
Open access
Sep 2026
Artificial intelligence-assisted lead optimization in drug discovery: bridging computational advances and translational challenges.
It is concluded that future progress will depend less on increasingly sophisticated algorithms than on trustworthy AI systems that improve scientific decision-making within iterative lead optimization workflows and ultimately enhance translational success in drug discovery.
F. A. Mohamed, A. M. K. El-sagheir
· Medicinal Chemistry Research · 0 citations