Sterically Controlled Chemoselective Synthesis of Chiral [3.3.1]-Bridged N-Heterocycles via Organocatalytic Asymmetric Multicomponent Dearomatization
Combining multicomponent reactions (MCRs) and catalytic asymmetric dearomatization (CADA) strategy in a tandem process to rapidly assemble valuable bridged N-heterocycles from indoles and other readily available materials remains extremely challenging with scarce reports. Herein, we report a chiral phosphoric acid (C...