Review
Jul 2026
Fourth-generation allosteric EGFR inhibitors: Structure-based scaffold analysis and SAR exploration.
It is established that allosteric EGFR inhibition represents a clinically viable strategy for addressing osimertinib resistance, with lead candidates ready for clinical translation.
Ibrahim Mohammed Hepishy, Mo'men Salem, A. El-Morsy et al.
· Bioorganic chemistry (Print) · 0 citations