Review
Open access
Aug 2026
Cysteine-targeting covalent inhibition: Recent trends and emerging strategies.
Design and chemistry principles of cysteine-targeting covalent inhibitors are addressed, with a focus on the diversity of electrophilic warheads currently used or under research, and established motifs are discussed alongside newfound warheads.
Mariana Castelôa, F. Borges, S. Benfeito et al.
· European journal of medicina... · 0 citations